Compile Data Set for Download or QSAR
Found 44 from National Institute of Industrial Technology
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)copy SMILEScopy InChI
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  0.580nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)copy SMILEScopy InChI
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu from recombinant RasGRP1 C1 domain (unknown origin) after 10 mins by scintillation counting analysis in presence of phosphat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]PDBu from recombinant human GFP-tagged RasGRP3 expressed in Escherichia coli BL21 after 5 mins by scintillation counting analysis...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017891(CHEMBL3289013)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017890(CHEMBL3289012)copy SMILEScopy InChI
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017892(CHEMBL3289014)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50017889(CHEMBL3289011)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-alpha after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Displacement of [3H]PDBu from recombinant human PKC-epsilon after 5 mins by scintillation counting analysis in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P270QKPubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241856(CHEMBL4097154)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241849(CHEMBL4070999)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241855(CHEMBL4075373)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50244449((E)-(2-(hydroxymethyl)-4-((1-methyl-1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241855(CHEMBL4075373)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241846(CHEMBL4069954)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241849(CHEMBL4070999)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241851(CHEMBL4099579)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241851(CHEMBL4099579)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241855(CHEMBL4075373)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241849(CHEMBL4070999)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241851(CHEMBL4099579)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241856(CHEMBL4097154)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241846(CHEMBL4069954)copy SMILEScopy InChI
Affinity DataKi:  119nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241856(CHEMBL4097154)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241850(CHEMBL4081576)copy SMILEScopy InChI
Affinity DataKi:  133nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241846(CHEMBL4069954)copy SMILEScopy InChI
Affinity DataKi:  257nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241850(CHEMBL4081576)copy SMILEScopy InChI
Affinity DataKi:  295nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241854(CHEMBL4066764)copy SMILEScopy InChI
Affinity DataKi:  301nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCepsilon (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241850(CHEMBL4081576)copy SMILEScopy InChI
Affinity DataKi:  504nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetRAS guanyl-releasing protein 1(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241854(CHEMBL4066764)copy SMILEScopy InChI
Affinity DataKi:  666nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from RasGRP1 (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation co...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institute of Industrial Technology

Curated by ChEMBL
LigandPNGBDBM50241854(CHEMBL4066764)copy SMILEScopy InChI
Affinity DataKi:  698nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from PKCalpha (unknown origin) in the presence of porcine brain phosphatidylserine by scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P62P2PubMed